Article(id=1322923389870022841, tenantId=1146029695717560320, journalId=1255847919539208197, issueId=1322923268038078806, articleNumber=null, orderNo=null, doi=10.13193/j.issn.1673-7717.2025.04.028, pmid=null, cstr=null, oa=null, hot=null, price=null, onlineType=0, articleFormat=0, articleType=null, articleTypeStr=null, receivedDate=null, receivedDateStr=null, revisedDate=null, revisedDateStr=null, acceptedDate=null, acceptedDateStr=null, onlineDate=1793339114873, onlineDateStr=2026-10-30, pubDate=1744214400000, pubDateStr=2025-04-10, doiRegisterDate=null, doiRegisterDateStr=null, onlineIssueDate=1793339114873, onlineIssueDateStr=2026-10-30, onlineJustAcceptDate=null, onlineJustAcceptDateStr=null, onlineFirstDate=null, onlineFirstDateStr=null, sourceXml=null, magXml=null, createTime=1793339114873, creator=13701087609, updateTime=1793339114873, updator=13701087609, issue=Issue{id=1322923268038078806, tenantId=1146029695717560320, journalId=1255847919539208197, year='2025', volume='43', issue='4', pageStart='1', pageEnd='258', issueExtLink='null', onlineDate='null', pubDate='1744214400000', pubDateStr='2025-04-10', beforeIssueId=null, nextIssueId=null, price=null, status=1, issueComplete=1, articleOrder=1, issueType=-1, specialIssue=0, createTime=1793339085826, creator='13701087609', updateTime=1793340586453, updator='13701087609', preIssue=null, nextIssue=null, articleTotal=null, ext={EN=IssueExt(id=1322929562572686061, tenantId=1146029695717560320, journalId=1255847919539208197, issueId=1322923268038078806, language=EN, specialIssueTitle=, coverIllustrator=null, specialIssueEditor=, specialIssueAbout=), CN=IssueExt(id=1322929562572686062, tenantId=1146029695717560320, journalId=1255847919539208197, issueId=1322923268038078806, language=CN, specialIssueTitle=, coverIllustrator=null, specialIssueEditor=, specialIssueAbout=)}, issueFiles=null, downloadFileDto=null}, startPage=176, endPage=180, ext={EN=ArticleExt(id=1322923391849734330, articleId=1322923389870022841, tenantId=1146029695717560320, journalId=1255847919539208197, language=EN, title=Quality Control Status and Predictive Analysis of Quality Markers of Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma), columnId=1256183361521967297, journalTitle=Chinese Archives of Traditional Chinese Medicine, columnName=Target on National Project, runingTitle=null, highlight=null, articleAbstract=

Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)contains various active ingredients,including flavonoids,phenylethanoid glycosides,organic acids and polysaccharides. Modern pharmacological studies indicate that Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)has pharmacological effects such as anti-inflammatory,antioxidant,anti-fatigue,anti-hypoxia,anti-aging,anticancer,hepatoprotective and symptom-alleviating properties in mild Alzheimer's disease. It also shows potential pharmacological effects in treating Parkinson's disease and severe depressive disorders,with promising application prospects. On the basis of summarizing the current status of quality control of Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)and understanding the concept of quality markers,this study predicted and analyzed the quality markers of Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)from eight aspects,including plant phylogeny,medicinal properties,medicinal efficacy,new medicinal uses,different compatibilities,measurability of chemical components,different harvesting periods and processing methods and different geographical origins,hoping to provide reference for establishing quality standards for Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma).

, authors=Jia HE, Meng’en YANG, Jingjing SHI, Mingsan MIAO, authorsList=Jia HE, Meng’en YANG, Jingjing SHI, Mingsan MIAO, authorCompany=null, correspAuthors=Mingsan MIAO, authorNote=null, correspAuthorsNote=null, copyrightStatement=null, copyrightOwner=null, extLink=null, articleAbsUrl=null, sourceXml=null, magXml=null, pdfUrl=null, pdf=null, pdfFileSize=null, pdfExtLink=null, richHtmlUrl=null, mobilePdfUrl=null, reviewReport=null, pdfFirstPage=null, abstractGraph=null, abstractGraphContent=null, abstractVideo=null, citation=null, cebUrl=null, magXmlContent=null, mapNumber=null, fund=null), CN=ArticleExt(id=1322923393170940093, articleId=1322923389870022841, tenantId=1146029695717560320, journalId=1255847919539208197, language=CN, title=红景天的质量控制现状及质量标志物预测分析, columnId=1256183362172142382, journalTitle=中华中医药学刊, columnName=国家项目点击, runingTitle=null, highlight=null, articleAbstract=

红景天中含有黄酮类、苯烷基苷类、有机酸类、多糖类等多种活性成分。现代药理研究表明,红景天具有抗炎、抗氧化、抗疲劳、抗缺氧、抗衰老、抗癌、保肝护肝、减缓轻度阿尔茨海默病症状以及具有潜在治疗帕金森病、重度抑郁病症的药理作用,且有良好的应用前景。在概括红景天质量控制现状以及理解质量标志物概念的基础上,从植物亲缘性、药性、药效、新的药效用途、不同配伍、化学成分的可测性、不同采收期及不同炮制方法、不同产地等8个方面对红景天的质量标志物进行了预测分析,以期为建立红景天中药材的质量标准提供参考。

, authors=贺嘉, 杨蒙恩, 史晶晶, 苗明三, authorsList=贺嘉, 杨蒙恩, 史晶晶, 苗明三, authorCompany=null, correspAuthors=苗明三, authorNote=

贺嘉(1999-),男,河南漯河人,硕士在读,研究方向:中药药理学。

, correspAuthorsNote=
苗明三(1965-),男,河南郑州人,教授,博士研究生导师,博士,研究方向:中药药理教学与研究。E-mail:。
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贺嘉(1999-),男,河南漯河人,硕士在读,研究方向:中药药理学。

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贺嘉(1999-),男,河南漯河人,硕士在读,研究方向:中药药理学。

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中药来源产地药用部位性味归经化学成分
大花红景天景天科红景天属中国西藏、云南西北部、四川西部根及根茎甘、苦、平归心、肝经红景天苷(Rhodiola Rosea)和大花红天素(Crenulatin)
狭叶红景天景天科红景天属西藏、云南、四川、新疆等地根茎微苦、涩、温归心、肺、大肠经红景天苷(Rhodiola Rosea)和酪醇(4-Hydroxyphenyl ethanol)
高山红景天景天科红景天属黑龙江、吉林全草甘、涩、平归心、肺、脾经红景天苷(Rhodiola Rosea)和没食子酸(Gallic acid)
), ArticleFig(id=1322923403505705186, tenantId=1146029695717560320, journalId=1255847919539208197, articleId=1322923389870022841, language=CN, label=表1, caption=

大花红景天与其他红景天的主要特征区别

, figureFileSmall=null, figureFileBig=null, tableContent=
中药来源产地药用部位性味归经化学成分
大花红景天景天科红景天属中国西藏、云南西北部、四川西部根及根茎甘、苦、平归心、肝经红景天苷(Rhodiola Rosea)和大花红天素(Crenulatin)
狭叶红景天景天科红景天属西藏、云南、四川、新疆等地根茎微苦、涩、温归心、肺、大肠经红景天苷(Rhodiola Rosea)和酪醇(4-Hydroxyphenyl ethanol)
高山红景天景天科红景天属黑龙江、吉林全草甘、涩、平归心、肺、脾经红景天苷(Rhodiola Rosea)和没食子酸(Gallic acid)
), ArticleFig(id=1322923405183426787, tenantId=1146029695717560320, journalId=1255847919539208197, articleId=1322923389870022841, language=EN, label=null, caption=null, figureFileSmall=null, figureFileBig=null, tableContent=
名称英文名称分子式文献
大花红天素CrenulatinC25H20O10[15]
酪醇4-Hydroxyphenyl ethanolC8H10O2[16]
红景天苷SalidrosideC14H20O7[17]
没食子酸Gallic acidC7H6O5[16]
咖啡酸3-(3,4-Dihydroxyphenyl)prop-2-enoic acidC9H8O4[16]
没食子酸乙酯Ethyl gallateC9H10O5[38]
芦丁RutinC27H30O16[41]
鞣花酸Ellagic acidC14H6O8[42]
络赛维RosavinC20H28O10[43]
草质素-7-O-鼠RhodioninC21H20O11[46]
李糖苷
草质素HerbacetinC15H10O7[50]
山柰酚KaempferolC15H10O6[50]
), ArticleFig(id=1322923405300867300, tenantId=1146029695717560320, journalId=1255847919539208197, articleId=1322923389870022841, language=CN, label=表2, caption=

红景天质量标志物预测

, figureFileSmall=null, figureFileBig=null, tableContent=
名称英文名称分子式文献
大花红天素CrenulatinC25H20O10[15]
酪醇4-Hydroxyphenyl ethanolC8H10O2[16]
红景天苷SalidrosideC14H20O7[17]
没食子酸Gallic acidC7H6O5[16]
咖啡酸3-(3,4-Dihydroxyphenyl)prop-2-enoic acidC9H8O4[16]
没食子酸乙酯Ethyl gallateC9H10O5[38]
芦丁RutinC27H30O16[41]
鞣花酸Ellagic acidC14H6O8[42]
络赛维RosavinC20H28O10[43]
草质素-7-O-鼠RhodioninC21H20O11[46]
李糖苷
草质素HerbacetinC15H10O7[50]
山柰酚KaempferolC15H10O6[50]
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红景天的质量控制现状及质量标志物预测分析
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贺嘉 , 杨蒙恩 , 史晶晶 , 苗明三
中华中医药学刊 | 国家项目点击 2025,43(4): 176-180
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中华中医药学刊 |国家项目点击 2025 , 43 (4) : 176 -180
红景天的质量控制现状及质量标志物预测分析
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贺嘉, 杨蒙恩, 史晶晶, 苗明三
作者信息
  • 河南中医药大学药学院,河南 郑州 450046
通讯作者:
苗明三(1965-),男,河南郑州人,教授,博士研究生导师,博士,研究方向:中药药理教学与研究。E-mail:。
作者简介:

贺嘉(1999-),男,河南漯河人,硕士在读,研究方向:中药药理学。

Quality Control Status and Predictive Analysis of Quality Markers of Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)
Jia HE, Meng’en YANG, Jingjing SHI, Mingsan MIAO
Affiliations
  • Henan University of Chinese Medicine, Zhengzhou 450046, Henan, China
出版时间: 2025-04-10 doi: 10.13193/j.issn.1673-7717.2025.04.028
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红景天中含有黄酮类、苯烷基苷类、有机酸类、多糖类等多种活性成分。现代药理研究表明,红景天具有抗炎、抗氧化、抗疲劳、抗缺氧、抗衰老、抗癌、保肝护肝、减缓轻度阿尔茨海默病症状以及具有潜在治疗帕金森病、重度抑郁病症的药理作用,且有良好的应用前景。在概括红景天质量控制现状以及理解质量标志物概念的基础上,从植物亲缘性、药性、药效、新的药效用途、不同配伍、化学成分的可测性、不同采收期及不同炮制方法、不同产地等8个方面对红景天的质量标志物进行了预测分析,以期为建立红景天中药材的质量标准提供参考。

红景天  /  质量控制  /  质量标志物

Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)contains various active ingredients,including flavonoids,phenylethanoid glycosides,organic acids and polysaccharides. Modern pharmacological studies indicate that Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)has pharmacological effects such as anti-inflammatory,antioxidant,anti-fatigue,anti-hypoxia,anti-aging,anticancer,hepatoprotective and symptom-alleviating properties in mild Alzheimer's disease. It also shows potential pharmacological effects in treating Parkinson's disease and severe depressive disorders,with promising application prospects. On the basis of summarizing the current status of quality control of Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)and understanding the concept of quality markers,this study predicted and analyzed the quality markers of Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)from eight aspects,including plant phylogeny,medicinal properties,medicinal efficacy,new medicinal uses,different compatibilities,measurability of chemical components,different harvesting periods and processing methods and different geographical origins,hoping to provide reference for establishing quality standards for Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma).

Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)  /  quality control  /  quality markers
贺嘉, 杨蒙恩, 史晶晶, 苗明三. 红景天的质量控制现状及质量标志物预测分析. 中华中医药学刊, 2025 , 43 (4) : 176 -180 . DOI: 10.13193/j.issn.1673-7717.2025.04.028
Jia HE, Meng’en YANG, Jingjing SHI, Mingsan MIAO. Quality Control Status and Predictive Analysis of Quality Markers of Hongjingtian(Rhodiolae Crenulatae Radix et Rhizoma)[J]. Chinese Archives of Traditional Chinese Medicine, 2025 , 43 (4) : 176 -180 . DOI: 10.13193/j.issn.1673-7717.2025.04.028
红景天基源为景天科红景天属植物大花红景天、高山红景天、圣地红景天、唐古特红景天等的根或根茎[1]。2020年版《中华人民共和国药典》收载品种为景天科植物大花红景天Rhodiola crenulata(Hook. f. et Thoms.)H. Ohba[2]。红景天入药始载于藏药著作《四部医典》[3],传统医书中将红景天列为药中上品[4]。红景天生于海拔2800~5600 m的山坡草地灌丛或石缝中,主要分布在西藏、云南、四川等地。红景天主要功效为益气活血,通脉平喘,用于气虚血瘀,胸痹心痛,中风偏瘫,倦怠气喘。现代药理研究发现,红景天中含有黄酮类、苯烷基苷类、有机酸类、多糖类等化合物,具有抗炎、抗氧化、抗疲劳、抗缺氧、抗衰老、抗癌、保肝护肝、减缓轻度阿尔茨海默病症状以及具有潜在治疗帕金森病、重度抑郁病症的药理活性[5]。本研究概括了红景天的质量控制现状,根据质量标志物(Quality marker,Q-Maker)的概念[6],对红景天潜在的质量标志物进行预测分析,以期为红景天质量标准的完善提供依据。
2020年版《中华人民共和国药典》一部记载了红景天的鉴别检查和含量测定,把红景天苷(Rhodiola Rosea)在红景天中的含量占比作为含量测定的标准,方法是通过高效液相色谱法(High performance liquid chromatography,HPLC)测定,红景天苷不得少于0.50%。但是仅将一种成分作为质量控制指标,不能全面展现红景天药材的品质。程益清等[7]使用高效液相色谱法对红景天中的红景天苷和酪醇(4-Hydroxyphenyl ethanol)成分进行含量测定,此方法高效可靠稳定性好,可作为红景天多种有效成分的含量测定方法,为红景天品质控制提供了参考。李志强等[8]用超高压液相色谱-三重四极杆串联飞行时间质谱法(Ultra-performance liquid chromatography-quadrupole time-of-flight/mass spectrometry,UPLC-Q-TOF/MS)对长鞭红景天提取物进行定性鉴别分析,鉴别出有机酚酸类、苯乙醇苷类、黄酮及萜类等36个化合物。李冲等[9]使用指纹图谱结合化学模式识别的方法分类鉴定红景天的品种,结果发现对长鞭红景天和四裂红景天有很好的区分效果,为控制红景天的质量提供了依据。马小东等[10]用超高效液相色谱法(Ultra-high-performance liquid chromatography,UHPLC)法同时测定唐古特红景天根中没食子酸(Gallic acid)、酪醇、红景天苷、没食子酸乙酯(Ethyl gallate)和对香豆酸(Cis-4-coumaric acid)的含量,为质量标志物的选择提供了参考。刘丹妮等[11]采用超高效液相色谱法同时测定蔷薇红景天中络塞维(Rosavin)、络塞琳(Rosarin)和络塞定(Rosiridin)的含量。邹亮等[12]采用HPLC-小粒径色谱柱法测定了红景天提取物中的红景天苷、酪醇和络赛维的含量。以上方法多以一种或一类成分对红景天进行质量控制的研究,有一定作用,但是中药化学成分复杂,且经过加工、炮制、提取、制剂、代谢等程序效应成分与原有成分已不太一致。因此,本研究结合红景天的最新质量研究现状从以下几个方面对红景天的质量标志物进行预测,为红景天的质量控制提供参考依据。
红景天成分复杂,需要从红景天种植、采收、炮制、制剂及代谢全过程进行把控,筛选质量标志物,在概括红景天质量控制现状以及理解质量标志物概念的基础上,从植物亲缘性、传统药性、传统药效、新的药效用途、不同配伍、化学成分的可测性、不同采收期及不同炮制方法、不同产地等8个方面对红景天的质量标志物进行了预测分析,以期为红景天的质量控制提供参考。
红景天是景天科红景天属植物,红景天属植物全世界约产90种,我国约有73种,另有2亚种和7变种[13],主要分布在东北、甘肃、新疆、四川、西藏及云贵等地区。景天科植物全世界共有34属超过1500种,中国有10属242种[14]。从植物亲缘学方面出发,景天科红景天属的植物很多,但是在药典中已经清楚地规定了红景天属用来入药的品种,并说明了其品质控制的标准。《中华人民共和国药典》明确指出红景天药材红景天苷所占比例应高于0.50%、醇浸出物不得少于22%。目前我国具有质量标准的药用红景天共有五种,分别为大花红景天、狭叶红景天、唐古红景天、长鞭红景天和高山红景天,宋霞等[15]使用气相色谱-串联质谱(Gas chromatography-tandem mass spectrometry,GC-MS/MS)建立了这5种红景天的指纹图谱并用化学模式识别,结果发现大花红天素(Crenulatin)、酪醇(4-Hydroxyphenyl ethanol)和红景天苷等成分指纹图谱出现明显差异,为不同红景天的主要差异成分,其中大花红天素为大花红景天的特异性成分。吕秀梅等[16]用高效液相色谱法同时测定大花红景天、狭叶红景天和长鞭红景天药材中没食子酸、红景天苷、酪醇、咖啡酸(Caffeic acid)、对香豆酸含量,结果发现不同品种红景天中化学成分含量存在较大差异,其中大花红景天红景天苷、没食子酸及咖啡酸含量最高,差异最明显。长白山地区同时存在高山红景天及易混淆的长白红景天,包文芳等[17]同时测定高山红景天和长白红景天中红景天苷含量,结果长白红景天中未检测出红景天苷。《中华人民共和国药典》记载的大花红景天与其他红景天的区别见表1。综上所述,可以将大花红天素、酪醇、红景天苷、没食子酸、咖啡酸作为红景天质量标志物的重要参考。
药性是中药理论必不缺少的一环,中药药性主要包括性味归经、升降浮沉、有毒无毒等。
张铁军等[18]认为药性物质基础的发现和确定有助于反映中药有效性的完整性,凸显中医药理论体系特点,可以帮助质量标志物的确定。红景天性寒味甘,归肺经。甘味药多用治正气虚弱、身体诸痛及调和药性、中毒解救等几个方面[19]。《素问·至真要大论篇》曰:“甘能补能缓”。甘味药化学成分以糖类、蛋白质、氨基酸类偏多[20-21]。林晓月等[22]优化了红景天多糖的制备工艺,并系统评价红景天多糖清除自由基的能力,研究结果表明红景天多糖具备抗氧化作用。王小雪等[23]发现归肺经中药主要化学成分包括黄酮类、挥发油类、苷类和萜类,这些成分具有抗菌、抗炎、抗病毒的作用,可以治疗感冒、咳喘等症状。综上所述,可以将糖类、蛋白质、氨基酸类、黄酮类、挥发油类、苷类和萜类作为红景天质量标志物的重要参考。
中药药效是中药治疗疾病性能的客观描述,是中医理论的核心理念[24]。2020版《中华人民共和国药典》记载红景天具有益气活血,通脉平喘的功效。《四部医典》中记载其功效为抗炎、清热、消肿。马莹慧等[25]的研究发现,红景天黄酮经过纯化后可显著抑制炎症因子(Tumor necrosis factor-alpha,TNF-α)的分泌,阻断炎症的发生。李英英等[26]探讨了有氧运动联合红景天口服液(主要成分为红景天苷、酪醇)对大鼠抗疲劳能力的影响。结果发现大鼠抗疲劳能力显著上升。潘梦之等[27]评价了红景天苷对脓毒症小鼠脾脏免疫细胞数量及功能的影响,发现红景天苷可显著改善脓毒症小鼠脾脏免疫功能。付金容等[28]研究了红景天苷对慢性间断性缺氧大鼠心肌炎症反应的影响,发现红景天苷可以抑制炎症反应,改善心功能。综上所述,可以将红景天黄酮、红景天苷、酪醇作为红景天质量标志物的重要参考依据。
现代研究表明红景天具有抗氧化、抗高原反应、抗肿瘤、抗衰老的作用。祁永章等[29]研究了红景天苷在高海拔地区干预大鼠创伤性慢性创面后对创面愈合的影响,结果发现红景天苷可以促进微血管生成,减轻组织损伤,加速创面愈合。叶刚等[30]通过动物实验研究发现云南红景天可以通过提高机体抗氧化和清除机体自由基能力而发挥延缓衰老作用。申洪娇等[31]探究了红景天苷对结肠癌细胞SW480增殖、凋亡和裸鼠移植瘤生长的影响,结果发现红景天苷具有抑制结肠癌细胞增殖、迁移、侵袭的作用。周通等[32]探索了红景天苷对胆囊癌细胞生物学行为的影响及其抗肿瘤的分子机制,发现红景天苷可能通过介导糖酵解效应和ERK/HIF-1α通路抑制胆囊癌细胞增殖、迁移和侵袭。综上所述,可以将红景天苷作为红景天质量标志物的重要参考依据。
中药一般具有多种功效,中药理论中可以通过复方配伍增加或增强药效,针对不同病证使用不同复方以达到治疗效果[33]。何鑫等[34]研究了人参鹿茸复方(人参、鹿茸、黄精、红景天)组方及单味药对小鼠体力疲劳的影响,结果发现红景天可以协同起到明显的抗疲劳作用。谭晓宇等[35]探究了灵芝红景天复方制剂对免疫低下小鼠免疫功能的影响,发现红景天可以显著增加免疫缺陷小鼠的免疫功能。钟壮聪等[36]研究了红景天虫草复方对短期高原训练后骨骼肌与大脑组织氧合作用影响,发现红景天可以有效预防高原训练后大脑组织总血红蛋白浓度、携氧血红蛋白与脱氧血红蛋白浓度下降的情况。付健阳等[37]研究了红景天、蛹虫草、大黄配伍(中药复方FF)对1型糖尿病大鼠肾脏的保护作用,红景天在组方中起到改善氧化应激水平等作用。李晶等[38]研究了红参和红景天配伍前后主要成分及抗疲劳活性的变化,结果配伍后抗疲劳效果增强,同时红景天成分没食子酸、红景天苷和没食子酸乙酯含量增加。综上所述,可以将抗疲劳、增强免疫、抗氧化、保护肾脏等有效成分及没食子酸、红景天苷和没食子酸乙酯作为红景天不同配方中的质量标志物的重要参考依据。
中药化学成分复杂,需要将易于检测且性质稳定的有效化成分作为质量标志物评价中药质量[39]。王金荣等[40]采用HPLC法对红景天中的有效成分没食子酸、红景天苷、酪醇进行含量测定。任卫合等[41]采用电感耦合等离子体发光光谱和高效液相色谱测定了红景天矿物元素及有效成分红景天苷、芦丁(Rutin)、没食子酸的含量,并分析了矿物元素的分布特征,结果发现硼(B)、铬(Cr)、锶(Sr)等元素含量与有效成分含量呈正相关。于然等[42]利用超高效液相色谱-串联质谱(Ultra-high-performance liquid chromatography-tandem mass spectrometry,UHPLCMS-QQQ)负离子检测模式同时测定红景天中红景天苷、酪醇、没食子酸和鞣花酸(Ellagic acid)的含量。综上所述,可以将红景天苷、没食子酸、酪醇、芦丁、鞣花酸及B、Cr、Sr等矿物元素作为红景天质量标志物的重要参考依据。
中药材的品质与其种植地与采收时间也密切相关,不同的采收期会导致中药材成分出现差异。强巴卓嘎等[43]对4种采收时期的西藏红景天不同部位中红景天苷、酪醇、络赛维进行分析,结果发现3种活性成分均在9月中下旬时含量达到最大。任艳艳等[44]对两个不同采收时间蔷薇红景天的红景天苷含量进行测定,结果发现8月采收的蔷薇红景天中红景天苷的含量比7月份高。中药炮制时,不同的炮制方法会对中药的化学成分造成不同影响,导致中药的性质和药效受到影响[45]。因此可以将炮制前后改变的化学成分作为红景天的质量标志物。王洋等[46]对34批不同红景天建立HPLC特征图谱,结果发现红景天素(Rhodiosin)、草质素-7-O-鼠李糖苷(Rhodionin)两个成分含量保留外表皮的大花红景天饮片比除去外表皮的更高。何宝佳等[47]用HPLC法测定不同炮制方法对红景天中红景天苷和酪醇的含量的变化,结果发现酒蒸品的红景天苷和酪醇含量明显升高。综上所述,可以将红景天苷、酪醇、络赛维、草质素-7-O-鼠李糖苷作为红景天质量标志物的重要参考依据。
中药材的产地也是质量控制的重要组成部分,同种药材不同产地也会影响到药材的品质。李霓冰等[48]用HPLC法测定了西藏、四川、云南、吉林、新疆等9个不同产地红景天中红景天苷的含量,结果发现西藏红景天中所含的红景天苷明显高于其他产地的红景天。时文娟等[49]用HPLC法测定新疆、四川、西藏等产地大花红景天中红景天苷和酪醇的含量,其中新疆红景天苷含量最高为1.25%,西藏红景天苷含量最低为0.58%,西藏酪醇含量最高为0.38%,四川酪醇含量最低为0.29%。张杰等[50]采用高效液相色谱-二级线性阵列检测器法(High Performance Liquid Chromatography with Diode Array Detector,HPLC-DAD)同时测定不同产地红景天中的Ternatumoside Ⅱ、红景天欧素、红景天宁、草质素(Herbacetin)、山柰酚(Kaempferol)、大花红景天素等成分,比较它们的差异性,结果表明不同来源及不同品种的红景天各成分差异显著。方勇[51]采用硫酸蒽酮法测定了6个不同产地红景天的多糖成分含量,结果发现高山红景天多糖含量最高为4.87%,四川大花红景天含量最低只有1.06%。综上所述,可以将红景天苷、酪醇、Ternatumoside Ⅱ、红景天欧素、红景天宁、草质素、山柰酚、大花红景天素、红景天多糖作为红景天质量标志物的重要参考依据。
红景天是我国传统中药材,红景天具备诸多功效,是疗效较好的补益药。红景天在我国主要分布在四川、西藏及云南等地域。目前红景天市场上品种混乱,质量参差不齐的现象仍然存在[52]。为保证临床安全有效用药,应当建立和完善科学的红景天的质量控制体系。本研究依据中药质量标志物的筛选原则从红景天植物亲缘学、药性、药效、新药效用途、配伍、可测化学成分、炮制前后化学成分的对比、不同采收期和产地等多方面对红景天的质量标志物进行预测分析。得出大花红天素、酪醇、红景天苷、没食子酸、咖啡酸、没食子酸乙酯、芦丁、鞣花酸、络赛维、草质素-7-O-鼠李糖苷、草质素、山柰酚等成分可作为红景天质量标志物的筛选对象(见表2及图1)。本文为红景天质量标志物的筛选与确定进行了探讨,以期为红景天质量标准的建立提供依据。
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2025年第43卷第4期
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doi: 10.13193/j.issn.1673-7717.2025.04.028
  • 首发时间:2026-10-30
  • 出版时间:2025-04-10
补充材料
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出版历史
基金
国家中医药管理局开放课题(GZYKJS-2022-040-1)
国家中医药管理局岐黄学者项目(国中医药人教函2022-6)
河南省豫药全产业链协同创新中心(豫科技〔2023〕175号)
河南省国际合作重点项目(豫财科〔2023〕16号)
作者信息
    河南中医药大学药学院,河南 郑州 450046

通讯作者:

苗明三(1965-),男,河南郑州人,教授,博士研究生导师,博士,研究方向:中药药理教学与研究。E-mail:。
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https://castjournals.cast.org.cn/joweb/zhzyyxk/CN/10.13193/j.issn.1673-7717.2025.04.028
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2种不同金属材料的力学参数
科
Family
属数
Number of
genus
种数
Number of
species
占总种数比例
Percentage of
total species (%)
属
Genus
种数
Number of
species
占总种数比例
Percentage of total
species (%)
鹅膏菌科Amanitaceae 2 11 5.26 鹅膏菌属 Amanita 10 4.78
小菇科 Mycenaceae 2 12 5.74 丝盖伞属 Inocybe 5 2.39
多孔菌科 Polyporaceae 8 14 6.70 蜡蘑属 Laccaria 5 2.39
红菇科 Russulaceae 3 23 11.00 小皮伞属 Marasmius 6 2.87
小菇属 Mycena 11 5.26
光柄菇属 Pluteus 5 2.39
红菇属 Russula 17 8.13
栓菌属 Trametes 5 2.39
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