Structure-activity relationship studies of 3,4-disubstitued indole-2-ketone derivatives identify a potent glutaminyl cyclase inhibitor with antitumor activity against breast cancer
aCollege of Food and Bioengineering, Xihua University, Chengdu 610039, China
bDepartment of Clinical Oncology, The University of Hong Kong-Shenzhen Hospital, Shenzhen 518053, China
cKey Laboratory of Drug Targeting and Drug Delivery System of Ministry of Education, West China School of Pharmacy, Sichuan University, Chengdu 610041, China
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